Helen Frankenthaler Foundation

NMBR BB1 receptor agonist

A2A receptor antagonist 2 | CAS 2767206-20-0 | AbMole BioScience

A2A receptor antagonist 2

Cat. No. M40667 All AbMole products are for research use only, cannot be used for human consumption.

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Quality Control & Documentation

  • Purity: >99.0%
  • COA
  • MSDS

Biological Activity

A2A receptor antagonist 2 is a potent, highly selective adenosine receptor A2A antagonist with an IC50 value of 8.3 nM.

Chemical Information

Molecular Weight 493.53 Formula C25H28FN7O3 CAS Number 2767206-20-0 Storage Powder -20°C 3 years; 4°C 2 years In solvent -80°C 6 months; -20°C 1 month

References

[1] W-T Shen et al. Eur Rev Med Pharmacol Sci. SCH58261, the antagonist of adenosine A2A receptor, alleviates cadmium-induced preeclampsia via sirtiun-1/hypoxia-inducible factor-1α pathway in rats

[2] Anup Masih et al. Neurosci Lett. Design and development of 1,3,5-triazine-thiadiazole hybrids as potent adenosine A2A receptor (A2AR) antagonist for benefit in Parkinson's disease

[3] Lei Chen et al. Mol Carcinog. Adenosine A2A receptor activation reduces brain metastasis via SDF-1/CXCR4 axis and protecting blood-brain barrier

[4] E Ongini et al. Farmaco. Selective adenosine A2A receptor antagonists

[5] T M Palmer et al. Mol Pharmacol. 125I-4-(2-[7-amino-2-[2-furyl][1,2,4]triazolo[2,3-a][1,3,5] triazin-5-yl-amino]ethyl)phenol, a high affinity antagonist radioligand selective for the A2a adenosine receptor

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Keywords: A2A receptor antagonist 2 supplier, Adenosine Receptor, inhibitors, activators All AbMole products are for research use only, cannot be used for human consumption or veterinary use. We do not provide products or services to individuals. Please comply with the intended use and do not use AbMole products for any other purpose.

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