1. GC72235 (Phenylac1,D-Tyr(Et)2,Lys6,Arg8,des-Gly9)-Vasopressin acetate (Phenylac1,D-Tyr(Et)2,Lys6,Arg8,des-Gly9)-Vasopressin is a potent vasopressin V1 receptor (VP V1R) antagonist.
2. GC66678 2-(3-Trifluoromethylphenyl)glycine hydrochloride 2-(3-Trifluoromethylphenyl)glycine hydrochloride is a precursor of substituted 2-acetamido-5-aryl-l, 2,4-triazolones. Substituted 2-acetamido-5-aryl-l, 2,4-triazolones are dual V1a/V2 receptor antagonists and can be used in cardiovascular disease research.
3. GC30764 Argipressin (Vasopressin) Arginine-vasopressin, as an important hormone in the regulation of plasma osmolality and blood volume/pressure, always is used in the treatment of septic shock and decompensated cirrhosis.
4. GC12194 Atosiban RW22164; RWJ22164 Atosiban is a mixed antagonist of oxytocin and vasopressin receptors. It effectively inhibits uterine contractions and prolongs pregnancy by competitively blocking oxytocin receptors on uterine smooth muscle.
5. GC39849 Atosiban acetate Atosiban acetate (RW22164 acetate;RWJ22164 acetate) is a nonapeptide competitive vasopressin/oxytocin receptor antagonist, and is a desamino-oxytocin analogue.
6. GC31295 Balovaptan (RG7314) RG7314 Balovaptan (RG7314) is a novel, orally active, selective, and blood-brain barrier-penetrating vasopressin 1a (V1a) receptor antagonist.
7. GA20807 Big Endothelin-1 (1-38), human Big Endothelin-1 (1-38), human is the precursor of endothelin-1.
8. GA20808 Big Endothelin-1 (1-39), porcine Big Endothelin-1 (1-39), porcine is the precursor of endothelin-1.
9. GC12627 Conivaptan HCl YM-087 Conivaptan (hydrochloride) is a non-peptide antagonist of vasopressin receptor, with Ki values of 0.48 and 3.04 nM for rat liver V1A receptor and rat kidney V2 receptor respectively.
10. GC12303 Desmopressin A vasopressin receptor agonist
11. GC11265 Desmopressin Acetate Desmopressin Acetate (DDAVP), a synthetic peptide analog of vasopressin, is a safe antidiuretic and hemostatic compound that acts as a selective agonist at the vasopressin V2 membrane receptor (V2R).
12. GC16591 d[Cha4]-AVP human vasopressin V1B receptor agonist
13. GC15154 d[Leu4,Lys8]-VP Selective vasopressin V1B receptor agonist
14. GC61959 D[LEU4,LYS8]-VP TFA D[LEU4,LYS8]-VP TFA is a selective agonist of vasopressin V1b receptor, with the Kis of 0.16 nM, 0.52 nM, and 0.1.38 nM for rat, human and mouse V1b receptor, respectively.
15. GC72087 F992 TFA F992 TFA is an antidiuretic peptide and vasopressin (antidiuretic hormone) analogue.
16. GC65415 Felypressin acetate Felypressin acetate (PLV-2 acetate) is a non-catecholamine vasoconstrictor and a vasopressin 1 agonist.
17. GC11991 L-371,257 human oxytocin (OT) receptor antagonist
18. GC32453 Lixivaptan (VPA-985) VPA-985, WAY-VPA-985 Lixivaptan (VPA-985) (VPA-985, WAY-VPA 985) is an orally active and selective vasopressin receptor V2 antagonist, with IC50 values of 1.2 and 2.3 nM for human and rat V2, respectively.
19. GC14880 Mozavaptan novel competitive vasopressin receptor antagonist
20. GC44247 Mozavaptan (hydrochloride) OPC 31260 Mozavaptan is a benzazepine derivative that antagonizes the binding of arginine vasopressin (AVP) to vasopressin receptors located in the liver (V1; IC50 = 1.2 μM) and kidney (V2; IC50 = 14 nM).
21. GC10622 OPC 21268 OPC 21268 (OPC-21268) is an orally effective, nonpeptide, vasopressin V1 receptor antagonist with an IC50 of 0.4 μM.
22. GC30890 RG7713 (RO5028442) RO5028442 RG7713 (RO5028442) (RO5028442) is a highly potent and selective Brain-Penetrant Vasopressin 1a (V1a) receptor antagonist with Kis of 1 nM (hV1a) and 39 nM (mV1a).
23. GC69875 Selepressin acetate FE 202158 acetate Selepressin (FE 202158) acetate is a selective vasopressin V1A receptor agonist. Selepressin acetate is an effective vasoconstrictor and can be used in the research of septic shock.
24. GC72171 SKF 100398 SKF 100398 (d(CH2)5Tyr(Et)VAVP), an arginine vasopressin (AVP) analogue, is a specific antagonist of the antidiuretic effect of exogenous and endogenous AVP.
25. GC12462 SR 49059 Relcovaptan vasopressin V1A receptor antagonist
26. GC38948 SRX246 SRX246 is a centrally penetrant vasopressin 1a (V1a) receptor antagonist.
27. GC50376 SSR 149415 SSR 149415 is a selective, non-peptide antagonist of the Vasopressin V1b Receptor.
28. GC50246 TASP 0390325 Potent and selective V1B receptor antagonist; orally bioavailable
29. GC32463 Terlipressin Terlipressin is a vasopressin analogue with potent vasoactive properties.
30. GC39830 Terlipressin acetate Glycylpressin, Remestyp A prodrug form of lysipressin
31. GC70580 Terlipressin diacetate Terlipressin diacetate is a vasopressin analogue with potent vasoactive properties.
32. GC15575 Tolvaptan OPC 41061 AVP V2-receptor antagonist
33. GC74398 Vasopressin Dimer (parallel) (TFA) Vasopressin Dimer (parallel) TFA is a parallel dimer of Vasopressin.
34. GC31475 WAY-151932 (VNA-932) VNA-932; WAY-VNA 932 WAY-151932 (VNA-932) is a vasopressin V2-receptor agonist with IC50 of 80.3 nM and 778 nM in human-V2 binding and V1a binding assay.
